SCHEMBL16639166

SCHEMBL16639166

CC(C)(C)[Si](OC[C@H]1OC[C@@H](n2ccc(NC(=O)c3ccccc3)nc2=O)S1)(c1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.46
RIN1 Q13671 1/20 0.46
POLB P06746 1/20 0.44
P2RY6 Q15077 2/20 0.43
P2RY14 Q15391 2/20 0.43
NT5E P21589 1/20 0.43
CYP3A4 P08684 2/20 0.36
HTT P42858 3/20 0.33
SMYD2 Q9NRG4 3/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 1/20 0.32
ALK Q9UM73 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.32
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13881302 1.00 ABL1 (0.46) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL9067177 0.92 ABL1 (0.36) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL9067623 0.92 ABL1 (0.36) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL9067175 0.92 ABL1 (0.36) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL9067499 0.92 ABL1 (0.36) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL13881212 0.91 ABL1 (0.48) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL13881301 0.91 ABL1 (0.48) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL3761289 0.85 ABL1 (0.52) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL3657470 0.85 ABL1 (0.52) ABL1RIN1POLBP2RY6P2RY14
SCHEMBL3658551 0.85 ABL1 (0.52) ABL1RIN1POLBP2RY6P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190839-B1 A PROCESS FOR CHIRAL RESOLUTION OF 2-SUBSTITUTED 4-SUBSTITUTED 1,3-OXATHIOLANES AVEXA LTD (AU) 2015-04-15 EP disclosed