SCHEMBL16644609

SCHEMBL16644609

CCOC(=O)c1cnc(NC2(c3ccccc3)CCN(C(=O)[C@H](c3ccccc3)C(C)C)CC2)nc1

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 19/20 0.74
HDAC1 Q13547 19/20 0.74
HDAC2 Q92769 19/20 0.74
HDAC6 Q9UBN7 19/20 0.74
VNN1 O95497 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16644391 1.00 HDAC3 (0.74) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL16644606 0.89 HDAC3 (0.77) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL16644353 0.89 HDAC3 (0.77) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL16644384 0.86 HDAC3 (0.66) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL16644352 0.85 HDAC3 (1.00) HDAC3HDAC1HDAC2HDAC6
SCHEMBL16632311 0.85 HDAC3 (1.00) HDAC3HDAC1HDAC2HDAC6
SCHEMBL16632310 0.85 HDAC3 (1.00) HDAC3HDAC1HDAC2HDAC6
SCHEMBL16644382 0.85 HDAC3 (0.70) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL16644356 0.83 HDAC3 (0.71) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL17832599 0.83 HDAC1 (0.62) HDAC3HDAC1HDAC2HDAC6VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015054474-A1 PYRIMIDINE HYDROXY AMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS ACETYLON PHARMACEUTICALS, INC. (US) 2015-04-16 WO disclosed