SCHEMBL16645582

SCHEMBL16645582

Cc1sc2nc(Cc3cccc(C#N)c3)cc(=O)n2c1C(N)=O

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 15/20 0.76
GRIN2A Q12879 15/20 0.76
GRIA2 P42262 7/20 0.76
IDH1 O75874 1/20 0.44
NLRP3 Q96P20 1/20 0.39
ADRA1D P25100 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636664 0.91 GRIN1 (0.78) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16636747 0.89 GRIN1 (0.84) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16637712 0.87 GRIN1 (0.75) GRIN1GRIN2AGRIA2IDH1
SCHEMBL16645606 0.87 GRIN1 (1.00) GRIN1GRIN2AGRIA2
SCHEMBL16636986 0.85 GRIN1 (0.69) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16637149 0.85 GRIN1 (0.68) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16645615 0.82 GRIN2A (0.63) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16645478 0.80 GRIN1 (0.77) GRIN1GRIN2AGRIA2
SCHEMBL16645472 0.80 GRIN1 (0.62) GRIN1GRIN2AGRIA2IDH1NLRP3
SCHEMBL16637396 0.79 GRIN2A (0.69) GRIN1GRIN2AGRIA2IDH1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052226-A1 THIAZOLOPYRIMIDINONES AS MODULATORS OF NMDA RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2015-04-16 WO disclosed