SCHEMBL16645719

SCHEMBL16645719

COC(=O)c1cccc2cn(-c3ccc4c(c3)OCCO4)nc12

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.53
ALDH1A1 P00352 4/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
NPC1 O15118 2/20 0.53
PKM P14618 1/20 0.53
PARP1 P09874 16/20 0.50
RAB9A P51151 1/20 0.50
POLB P06746 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
TP53 P04637 1/20 0.46
KMT2A Q03164 1/20 0.46
PARP2 Q9UGN5 10/20 0.46
PARP3 Q9Y6F1 10/20 0.46
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635316 0.85 PARP1 (0.63) PARP1PARP2PARP3
SCHEMBL16645833 0.83 PARP1 (0.60) PARP1PARP2PARP3
SCHEMBL16645834 0.83 PARP1 (0.60) PARP1PARP2PARP3
SCHEMBL16645829 0.83 PARP1 (0.60) PARP1PARP2PARP3
SCHEMBL16645831 0.81 PARP1 (0.61) PARP1PARP2PARP3
SCHEMBL16635490 0.81 PARP1 (0.61) PARP1PARP2PARP3
SCHEMBL2265110 0.79 PARP1 (0.71) ALDH1A1PARP1MAPTKMT2APARP2
SCHEMBL2265978 0.79 PARP1 (0.47) PARP1PARP2PARP3
SCHEMBL16645828 0.79 PARP1 (0.63) PARP1PARP2PARP3
SCHEMBL1422526 0.79 PARP1 (0.68) ALDH1A1PARP1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051766-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY (ADP-RIBOSE) POLYMERASE INHIBITORS BETTA PHARMACEUTICALS CO., LTD (CN) 2015-04-16 WO disclosed