SCHEMBL16645934

SCHEMBL16645934

Cc1sc2nc(Cc3cccc(Cl)c3F)c(F)c(=O)n2c1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.42
GRIN2A Q12879 6/20 0.42
GRIA2 P42262 4/20 0.42
CD38 P28907 1/20 0.39
PCSK9 Q8NBP7 1/20 0.35
GRM4 Q14833 2/20 0.34
CFD P00746 1/20 0.34
P2RX7 Q99572 4/20 0.34
TRPA1 O75762 1/20 0.34
AADAT Q8N5Z0 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
GPR52 Q9Y2T5 1/20 0.33
CHRM4 P08173 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636982 0.86 GRIN1 (0.58) GRIN1GRIN2AGRIA2GRM4P2RX7
SCHEMBL16645938 0.86 GRIN1 (0.55) GRIN1GRIN2AGRIA2CD38P2RX7
SCHEMBL16645813 0.86 GRIN1 (0.41) GRIN1GRIN2AGRIA2
SCHEMBL16645466 0.75 GRIN1 (0.61) GRIN1GRIN2AGRIA2CD38P2RX7
SCHEMBL16645803 0.75 GRIN1 (0.46) GRIN1GRIN2AGRIA2
SCHEMBL16645600 0.75 GRIN1 (0.62) GRIN1GRIN2AGRIA2
SCHEMBL16645945 0.74 GRIN1 (0.43) GRIN1GRIN2AGRIA2
SCHEMBL17958237 0.73 GRIN1 (0.73) GRIN1GRIN2AGRIA2
SCHEMBL17958254 0.73 GRIN1 (0.56) GRIN1GRIN2AGRIA2
SCHEMBL17958250 0.73 GRIN1 (0.66) GRIN1GRIN2AGRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052226-A1 THIAZOLOPYRIMIDINONES AS MODULATORS OF NMDA RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2015-04-16 WO disclosed