SCHEMBL16649356

SCHEMBL16649356

Nc1ccc(OC(F)(F)F)c(C23COCCC2CSC(NC(=O)O)=N3)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.57
KCNH2 Q12809 3/20 0.41
CYP2D6 P10635 1/20 0.41
BACE2 Q9Y5Z0 3/20 0.34
WNT3A P56704 1/20 0.33
EPHX2 P34913 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3298246 1.00 BACE1 (0.57) BACE1KCNH2CYP2D6BACE2WNT3A
SCHEMBL7918201 0.89 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2WNT3A
SCHEMBL9913099 0.89 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2WNT3A
SCHEMBL7918182 0.89 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2WNT3A
SCHEMBL3779202 0.86 BACE1 (0.40) BACE1KCNH2BACE2WNT3AEPHX2
SCHEMBL3779198 0.86 BACE1 (0.40) BACE1KCNH2BACE2WNT3AEPHX2
SCHEMBL3307012 0.86 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2
SCHEMBL3304092 0.86 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2
SCHEMBL3302948 0.86 BACE1 (0.53) BACE1KCNH2CYP2D6BACE2
SCHEMBL1935243 0.82 BACE1 (0.54) BACE1KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2332943-B1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R&D MAN CO LTD (JP) 2015-04-22 EP disclosed