SCHEMBL16655832

SCHEMBL16655832

C=CC(=O)Nc1cc(CCN)ccc1Nc1cc(N(C)C(=O)Nc2c(Cl)c(OC)cc(OC)c2Cl)ncn1

nearest known ligand 0.86

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 17/20 0.86
FGFR2 P21802 2/20 0.76
FGFR3 P22607 2/20 0.76
FGFR4 P22455 3/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655985 0.94 FGFR1 (0.90) FGFR1FGFR2FGFR3FGFR4
SCHEMBL16659492 0.92 FGFR1 (1.00) FGFR1FGFR2FGFR3FGFR4
SCHEMBL18373850 0.92 FGFR1 (0.88) FGFR1FGFR2FGFR3FGFR4
SCHEMBL16654878 0.92 FGFR1 (1.00) FGFR1FGFR2FGFR3FGFR4
SCHEMBL16659432 0.91 FGFR1 (1.00) FGFR1FGFR2FGFR3FGFR4
SCHEMBL17728854 0.91 FGFR1 (1.00) FGFR1FGFR2FGFR3FGFR4
SCHEMBL16659468 0.91 FGFR1 (1.00) FGFR1FGFR2FGFR3FGFR4
SCHEMBL16659441 0.89 FGFR1 (0.94) FGFR1FGFR2FGFR3FGFR4
Trifluoroacetic Acid SCHEMBL17728863 0.89 FGFR1 (0.92) FGFR1FGFR2FGFR3FGFR4
SCHEMBL28096901 0.88 FGFR1 (0.79) FGFR1FGFR2FGFR3FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057943-A1 PYRIMIDINE FGFR4 INHIBITORS Eisai R&D Management Co., Ltd. (JP) 2016-08-24 EP disclosed
WO-2015057938-A1 PYRIMIDINE FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed