SCHEMBL16656140

SCHEMBL16656140

C=Cc1c(OC)cncc1OCc1cccnc1-c1ccnn1C(C)C

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C8 P10632 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
PDE1B Q01064 5/20 0.33
SGMS2 Q8NHU3 1/20 0.31
PDE1A P54750 4/20 0.31
PDE1C Q14123 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15065328 0.91 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL16656139 0.89 CYP1A2 (0.65) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL16072988 0.86 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL15066166 0.82 CYP1A2 (0.68) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL26110658 0.82 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL15068330 0.82 CYP1A2 (0.79) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL30077912 0.82 CYP1A2 (0.79) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL15065951 0.82 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL16671919 0.81 CYP1A2 (0.82) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL20192060 0.81 CYP1A2 (0.63) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9012450-B2 Substituted heteroaryl aldehyde compounds and methods for their use in increasing tissue oxygenation GLOBAL BLOOD THERAPEUTICS, INC. (US) 2015-04-21 US disclosed