SCHEMBL16659604

SCHEMBL16659604

C=CC(=O)Nc1cc(C(=O)N2CCN(C)CC2)ccc1Nc1cc(N(C)C(=O)Nc2cc(OC)cc(OC)c2Cl)ncn1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 15/20 0.83
FGFR4 P22455 4/20 0.72
FGFR3 P22607 3/20 0.63
FGFR2 P21802 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16659469 0.91 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL582750 0.86 FGFR3 (0.80) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659464 0.84 FGFR4 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659450 0.84 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL19732275 0.82 FGFR1 (0.84) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659504 0.82 FGFR4 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659425 0.81 FGFR4 (0.77) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659489 0.80 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL374467 0.78 FGFR3 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16665249 0.78 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015057938-A1 PYRIMIDINE FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed