SCHEMBL16664340

SCHEMBL16664340

NC1=N[C@@]2(c3cc(NC(=O)c4ccc(OC(F)F)cn4)ccc3F)COCCC2CS1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 1.00
KCNH2 Q12809 4/20 1.00
CYP2D6 P10635 2/20 1.00
BACE2 Q9Y5Z0 4/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3298238 1.00 BACE1 (1.00) BACE1KCNH2CYP2D6BACE2
SCHEMBL3298235 1.00 BACE1 (1.00) BACE1KCNH2CYP2D6BACE2
SCHEMBL8032820 0.92 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL2620250 0.92 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL3773260 0.92 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL9913173 0.91 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2
SCHEMBL7925082 0.91 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2
SCHEMBL16649481 0.91 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2
SCHEMBL16649482 0.91 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2
SCHEMBL3305562 0.90 BACE1 (0.82) BACE1KCNH2CYP2D6BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2332943-B1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R&D MAN CO LTD (JP) 2015-04-22 EP disclosed