SCHEMBL16664346

SCHEMBL16664346

NC1=N[C@@]2(c3cc(NC(=O)c4ccc(OC(F)F)cn4)ccc3F)COC[C@@H](F)C2CS1

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.75
KCNH2 Q12809 3/20 0.75
CYP2D6 P10635 2/20 0.75
BACE2 Q9Y5Z0 5/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1933972 1.00 BACE1 (0.75) BACE1KCNH2CYP2D6BACE2
SCHEMBL12557787 0.94 BACE1 (0.67) BACE1KCNH2CYP2D6BACE2
SCHEMBL1935180 0.90 BACE1 (0.61) BACE1KCNH2CYP2D6BACE2
SCHEMBL2620250 0.90 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL3773260 0.90 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL8032820 0.90 BACE1 (0.86) BACE1KCNH2CYP2D6BACE2
SCHEMBL16664344 0.88 BACE1 (0.70) BACE1KCNH2CYP2D6BACE2
SCHEMBL1935621 0.88 BACE1 (0.70) BACE1KCNH2CYP2D6BACE2
SCHEMBL7922912 0.88 BACE1 (0.70) BACE1KCNH2CYP2D6BACE2
SCHEMBL9913408 0.88 BACE1 (0.70) BACE1KCNH2CYP2D6BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2332943-B1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE EISAI R&D MAN CO LTD (JP) 2015-04-22 EP disclosed