SCHEMBL16664800

SCHEMBL16664800

CN(I)C(=O)[C@H]1CC[C@@H](OS(C)(=O)=O)[C@H](NC(=O)OC(C)(C)C)C1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.37
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36
KDM1A O60341 2/20 0.33
CTSK P43235 2/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10015600 0.91 BTK (0.39) BTKMAOBMAOAKDM1ACTSK
SCHEMBL10063105 0.87 MAOB (0.42) BTKMAOBMAOAKDM1ACTSK
SCHEMBL10476741 0.84 BTK (0.53) BTKMAOBMAOAKDM1ACTSK
SCHEMBL2712349 0.84 BTK (0.53) BTKMAOBMAOAKDM1ACTSK
SCHEMBL2712346 0.84 BTK (0.53) BTKMAOBMAOAKDM1ACTSK
SCHEMBL2709392 0.84 BTK (0.53) BTKMAOBMAOAKDM1ACTSK
SCHEMBL16664839 0.83 BTK (0.43) BTKMAOBMAOAKDM1ACTSK
SCHEMBL10063319 0.82 BTK (0.39) BTKMAOBMAOAKDM1ACTSK
SCHEMBL17472894 0.80 BTK (0.38) BTKMAOBMAOAKDM1ACTSK
SCHEMBL17437659 0.80 CA12 (0.36) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2407450-B1 Method for producing optically active diamine derivative DAIICHI SANKYO CO LTD (JP) 2015-04-22 EP disclosed