SCHEMBL16665256

SCHEMBL16665256

C=CC(=O)Nc1cccc(Nc2cc(N(C)C(=O)Nc3c(Cl)c(OC)cc(OC)c3Cl)ncn2)c1

nearest known ligand 0.77

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 14/20 0.77
FGFR4 P22455 4/20 0.77
FGFR3 P22607 3/20 0.77
FGFR2 P21802 1/20 0.77
CYP3A4 P08684 2/20 0.72
CYP2C19 P33261 2/20 0.72
CYP2C9 P11712 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16665288 0.87 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL17740756 0.87 FGFR4 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659606 0.87 FGFR2 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659436 0.86 FGFR1 (0.89) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16654398 0.86 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659401 0.86 FGFR1 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16659421 0.85 FGFR4 (0.88) FGFR1FGFR4FGFR3FGFR2
SCHEMBL16655616 0.85 FGFR4 (1.00) FGFR1FGFR4FGFR3FGFR2
SCHEMBL374485 0.83 FGFR3 (1.00) FGFR1FGFR4FGFR3FGFR2CYP3A4
SCHEMBL17856981 0.83 FGFR4 (0.62) FGFR1FGFR4FGFR3FGFR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015057963-A1 FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed