SCHEMBL16665267

SCHEMBL16665267

C=CC(=O)Nc1ccccc1Nc1cc(OCc2ccccc2)ccn1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 13/20 0.50
EGFR P00533 2/20 0.48
ERBB2 P04626 1/20 0.48
FGFR1 P11362 4/20 0.47
FGFR3 P22607 3/20 0.47
FGFR2 P21802 2/20 0.47
BTK Q06187 1/20 0.46
MAPK3 P27361 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CTSV O60911 1/20 0.43
CTSL P07711 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16665334 0.85 GCK (0.54) FGFR4EGFRERBB2FGFR1FGFR3
SCHEMBL16665247 0.79 FGFR4 (0.48) FGFR4EGFRFGFR1FGFR3FGFR2
SCHEMBL16665246 0.79 FGFR4 (0.56) FGFR4FGFR1FGFR3FGFR2MAPK3
SCHEMBL16665335 0.79 FGFR4 (0.59) FGFR4FGFR1FGFR3FGFR2MAPK3
SCHEMBL16665266 0.78 FGFR4 (0.54) FGFR4EGFRFGFR1FGFR3FGFR2
SCHEMBL16665336 0.78 FGFR4 (0.55) FGFR4FGFR1FGFR3FGFR2MAPK3
SCHEMBL26697665 0.77 MEN1 (0.59) MEN1KMT2ACTSVCTSL
SCHEMBL16665302 0.77 MAPK3 (0.50) FGFR4FGFR1FGFR3FGFR2MAPK3
SCHEMBL16665297 0.76 MAPK3 (0.49) FGFR4MAPK3
SCHEMBL16665248 0.76 GCK (0.50) FGFR4EGFRFGFR1FGFR3FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015057963-A1 FGFR4 INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-04-23 WO disclosed
US-20140107118-A1 Novel Heterocyclic Derivatives and Their Use in the Treatment of Neurological Disorders NOVARTIS AG (CH) 2014-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140107118-A1 Novel Heterocyclic Derivatives and Their Use in the Treatment of Neurological Disorders BACE2, BACE1, PSEN2 FGFR4 2244/4885EGFR 2424/4885ERBB2 621/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.