SCHEMBL16672212

SCHEMBL16672212

FC1(F)CNc2cc(Nc3nccn4nc(Nc5cccc(C(F)(F)F)c5)nc34)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 7/20 0.43
PTK2 Q05397 7/20 0.43
CLK1 P49759 1/20 0.39
CLK2 P49760 1/20 0.39
DYRK1A Q13627 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
JAK3 P52333 6/20 0.38
AURKA O14965 2/20 0.38
GRM4 Q14833 1/20 0.37
CTSC P53634 5/20 0.37
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
IDH2 P48735 2/20 0.36
CDK1 P06493 1/20 0.36
PRKCA P17252 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23034 0.86 JAK3 (0.48) JAK2PTK2CLK1CLK2DYRK1A
SCHEMBL23696 0.83 AURKA (0.52) JAK2PTK2JAK3AURKAGRM4
SCHEMBL24629 0.80 IDH2 (0.57) JAK2PTK2JAK3AURKACTSC
SCHEMBL23189 0.80 IDH2 (0.57) JAK2PTK2JAK3AURKACTSC
SCHEMBL24034 0.78 IDH2 (0.47) JAK2PTK2JAK3AURKACTSC
SCHEMBL24622 0.78 IDH2 (0.47) JAK2PTK2JAK3AURKACTSC
SCHEMBL23674 0.78 IDH2 (0.47) JAK2PTK2JAK3AURKACTSC
SCHEMBL21053 0.75 JAK3 (0.49) JAK2PTK2JAK3
SCHEMBL24621 0.75 MAPT (0.48) JAK2PTK2JAK3AURKAKDR
SCHEMBL23984 0.75 MAPT (0.48) JAK2PTK2JAK3AURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9023851-B2 Triazolopyrazine derivatives MERCK PATENT GMBH (DE) 2015-05-05 US claimed