SCHEMBL16690709

SCHEMBL16690709

COC(=O)c1ccc(C(=O)c2c(C)ccc(F)c2F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
CA7 P43166 1/20 0.46
NOTUM Q6P988 1/20 0.44
MAPT P10636 7/20 0.44
KMT2A Q03164 4/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
MEN1 O00255 3/20 0.44
HTT P42858 2/20 0.44
MAPK1 P28482 1/20 0.44
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31246136 0.84 CA12 (0.44) TDP1CA1CA2CA12CA9
SCHEMBL16690694 0.84 TDP1 (0.47) TDP1CA1CA2CA12CA9
SCHEMBL18044465 0.84 CA1 (0.50) TDP1CA1CA2CA12CA9
SCHEMBL18044458 0.83 CA1 (0.47) TDP1CA1CA2CA12CA9
SCHEMBL8480830 0.77 EGFR (0.45) TDP1CA1CA2CA12CA9
SCHEMBL20709025 0.76 MAPT (0.44) TDP1CA1CA2CA12CA9
SCHEMBL3518044 0.75 CA12 (0.48) TDP1CA1CA2CA12CA9
SCHEMBL2337244 0.74 CA1 (0.70) TDP1CA1CA2CA12CA9
SCHEMBL3205636 0.74 CA12 (0.44) TDP1CA1CA2CA12CA9
SCHEMBL1495863 0.74 HDAC1 (0.62) TDP1CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015062555-A1 COMPOUND HAVING HIGHER INHIBITION OF PROTEIN KINASE G ACTIVITY AND PREPARATION METHOD THEREFOR 天津键凯科技有限公司 2015-05-07 WO disclosed