SCHEMBL16695803

SCHEMBL16695803

Cc1ncc2[nH]c(=O)c3ccccc3n12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.54
CYP1A2 P05177 2/20 0.54
HPGD P15428 2/20 0.43
CYP2C9 P11712 1/20 0.43
LCK P06239 1/20 0.41
PRKACA P17612 1/20 0.41
CSNK2A2 P19784 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
GSK3B P49841 1/20 0.41
CSNK2B P67870 1/20 0.41
CSNK2A1 P68400 1/20 0.41
DYRK1A Q13627 1/20 0.41
CSNK2A3 Q8NEV1 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
HIF1A Q16665 1/20 0.40
CHEK1 O14757 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31515754 0.89 PARP1 (0.47) PARP1CYP1A2HPGDCYP2C9LCK
SCHEMBL31515706 0.81 PARP1 (0.45) PARP1CYP1A2HPGDLCKPRKACA
SCHEMBL15714749 0.77 PARP1 (0.53) PARP1CYP1A2HPGDCYP2C9LCK
SCHEMBL15083751 0.74 PARP1 (0.47) PARP1CYP1A2HPGDCYP2C9LCK
SCHEMBL11265442 0.72 KDM4E (0.44) HPGDLCKKDM4EALDH1A1CHEK1
SCHEMBL15887033 0.72 LCK (0.42) CYP1A2HPGDLCKKDM4EALDH1A1
SCHEMBL22045220 0.71 LCK (0.55) PARP1CYP1A2HPGDCYP2C9LCK
SCHEMBL22045317 0.70 CDC25B (0.54) PARP1CYP1A2LCKPRKACACSNK2A2
SCHEMBL29792766 0.70 PARP1 (1.00) PARP1CYP1A2RAB9A
SCHEMBL16695791 0.70 PARP1 (1.00) PARP1CYP1A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9708332-B2 Respiratory syncytial virus inhibitors MEDIVIR AB (SE) 2017-07-18 US disclosed
US-9708332-B2 Respiratory syncytial virus inhibitors MEDIVIR AB (SE) 2017-07-18 US disclosed
WO-2015065338-A1 QUINAZOLINE BASED RESPIRATORY SYNCYTIAL VIRUS INHIBITORS MEDIVIR AB (SE) 2015-05-07 WO disclosed