SCHEMBL16696136

SCHEMBL16696136

CC(C)CCn1c(Cn2c(=O)n(C3COC3)c3ccncc32)nc(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.50
TNKS O95271 1/20 0.36
OPRL1 P41146 5/20 0.36
CYP2D6 P10635 1/20 0.36
PDE5A O76074 1/20 0.35
ALDH1A1 P00352 3/20 0.35
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
OPRM1 P35372 3/20 0.34
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
PLK1 P53350 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
GRM4 Q14833 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16696137 0.93 CYP3A4 (0.49) CYP3A4TNKSOPRL1CYP2D6PDE5A
SCHEMBL16696088 0.92 CYP3A4 (0.59) CYP3A4TNKSOPRL1CYP2D6PDE5A
SCHEMBL16696058 0.92 CYP3A4 (0.53) CYP3A4TNKSOPRL1CYP2D6PDE5A
SCHEMBL16696115 0.87 CYP3A4 (0.46) CYP3A4TNKSOPRL1CYP2D6OPRM1
SCHEMBL9978093 0.87 CYP3A4 (0.49) CYP3A4TNKSOPRL1CYP2D6TSHR
SCHEMBL9977932 0.87 CYP3A4 (0.54) CYP3A4TNKSOPRL1CYP2D6TSHR
SCHEMBL16696052 0.86 CYP3A4 (0.49) CYP3A4TNKSOPRL1CYP2D6PDE5A
SCHEMBL16696071 0.84 CYP3A4 (0.56) CYP3A4TNKSOPRL1CYP2D6OPRM1
SCHEMBL16696092 0.83 OPRL1 (0.48) CYP3A4OPRL1CYP2D6PDE5AALDH1A1
SCHEMBL9978054 0.82 CYP3A4 (0.44) CYP3A4TNKSOPRL1CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015065336-A1 RESPIRATORY SYNCYTIAL VIRUS INHIBITORS MEDIVIR AB (SE) 2015-05-07 WO disclosed