SCHEMBL16701353

SCHEMBL16701353

CCCCCCCc1c(N)nc(N)nc1-c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.53
PPARA Q07869 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TLR8 Q9NR97 7/20 0.46
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
CYP2D6 P10635 2/20 0.42
HRH3 Q9Y5N1 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYP2A6 P11509 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
GBA1 P04062 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12495536 0.88 ADORA2A (0.50) DHFRPPARATDP1L3MBTL1TLR8
SCHEMBL12496398 0.84 ADORA2A (0.57) DHFRPPARATDP1L3MBTL1TLR8
SCHEMBL12496119 0.83 ADORA2A (0.49) DHFRPPARATDP1L3MBTL1TLR8
SCHEMBL12496114 0.82 TLR8 (0.46) PPARATDP1L3MBTL1TLR8ADORA2A
SCHEMBL12496127 0.80 KDM4E (0.48) PPARATLR8ADORA2AADORA1CYP2D6
SCHEMBL12496003 0.79 CYP3A4 (0.50) DHFRPPARATLR8ADORA2AADORA1
SCHEMBL12495799 0.79 ADORA2A (0.46) PPARATDP1TLR8ADORA2AADORA1
SCHEMBL21313209 0.78 CYP2A6 (0.48) PPARAL3MBTL1TLR8ADORA2AADORA1
SCHEMBL21313265 0.78 ADORA2A (0.46) PPARATDP1L3MBTL1TLR8ADORA2A
SCHEMBL16223070 0.78 CYP3A4 (0.50) PPARATDP1L3MBTL1TLR8ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069752-A9 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-07-09 WO disclosed
WO-2015069752-A1 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-05-14 WO disclosed