SCHEMBL16705122

SCHEMBL16705122

COCCNC(=O)c1sc(N2CCOCC2)c(C#N)c1-c1ccc(Cl)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.52
MTOR P42345 2/20 0.52
ALPL P05186 1/20 0.43
KMT2A Q03164 4/20 0.41
EGFR P00533 1/20 0.41
CDK2 P24941 1/20 0.41
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13597970 0.92 PIK3CA (0.52) PIK3CAMTORKMT2AEGFRCDK2
SCHEMBL8006058 0.91 PIK3CA (0.54) PIK3CAMTORKMT2AEGFRCDK2
SCHEMBL8008169 0.91 PIK3CA (0.50) PIK3CAMTORKMT2AEGFRCDK2
SCHEMBL8005712 0.90 PIK3CA (0.53) PIK3CAMTOREGFRCDK2MAPT
SCHEMBL8008105 0.90 PIK3CA (0.53) PIK3CAMTOREGFRCDK2MAPK1
SCHEMBL7996257 0.90 PIK3CA (0.55) PIK3CAMTORALPLEGFRCDK2
SCHEMBL8006078 0.90 PIK3CA (0.56) PIK3CAMTORKMT2AEGFRCDK2
SCHEMBL8008138 0.90 PIK3CA (0.52) PIK3CAMTOREGFRCDK2ALDH1A1
SCHEMBL1552132 0.90 PIK3CA (0.55) PIK3CAMTOREGFRCDK2ALDH1A1
SCHEMBL13597813 0.90 PIK3CA (0.54) PIK3CAMTOREGFRCDK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9029411-B2 Thiophenes and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-05-12 US disclosed