SCHEMBL16705270

SCHEMBL16705270

CCOC(=O)Cn1cnc2c(N)nc(NC)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.46
CCNB1 P14635 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
TMIGD3 P0DMS9 4/20 0.45
ADORA2A P29274 4/20 0.45
ADORA1 P30542 4/20 0.45
ADORA2B P29275 2/20 0.45
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
TLR9 Q9NR96 1/20 0.41
HPRT1 P00492 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
JAK3 P52333 1/20 0.40
MITF O75030 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10047134 0.87 ADORA2A (0.51) CDK1CCNB1CCNE1CDK2TMIGD3
SCHEMBL431825 0.85 CDK1 (0.61) CDK1CCNB1CCNE1CDK2KDM4E
SCHEMBL10047144 0.85 ADORA2A (0.52) CDK1CDK2TMIGD3ADORA2AADORA1
SCHEMBL10047141 0.84 ADORA2A (0.51) CDK1CDK2TMIGD3ADORA2AADORA1
SCHEMBL10072757 0.83 ADORA2A (0.48) CDK1CDK2TMIGD3ADORA2AADORA1
SCHEMBL10047089 0.81 ADORA2A (0.40) CDK1CCNB1CCNE1CDK2TMIGD3
SCHEMBL611356 0.80 CDK1 (0.43) CDK1CDK2TMIGD3ADORA2AADORA1
SCHEMBL29728010 0.79 ADORA2A (0.60) ADORA2AADORA1ADORA2BLMNAEP300
SCHEMBL14611764 0.79 CDK1 (0.48) CDK1CCNB1CCNE1CDK2KDM4E
SCHEMBL1565498 0.79 ADORA2A (0.60) ADORA2AADORA1ADORA2BLMNAEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268607-B9 PEPTIDE NUCLEIC ACID DERIVATIVES WITH GOOD CELL PENETRATION AND STRONG AFFINITY FOR NUCLEIC ACID CTI BIO (KR) 2015-05-13 EP disclosed