SCHEMBL1670655

SCHEMBL1670655

O=C(NC1(C(=O)O)CC1)c1cccc(C2(NC(=O)c3cncc4c3cnn4-c3ccc(F)cc3)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.61
KCNH2 Q12809 2/20 0.61
ADRB1 P08588 1/20 0.61
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670713 0.91 CCR1 (0.61) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670417 0.91 CCR1 (0.66) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670699 0.89 CCR1 (0.66) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1672943 0.88 CCR1 (0.65) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670697 0.87 CCR1 (0.70) CCR1KCNH2ADRB1CYP3A4
SCHEMBL12799627 0.87 CCR1 (0.61) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1670486 0.87 CCR1 (0.65) CCR1KCNH2ADRB1CYP3A4
SCHEMBL12799605 0.86 CCR1 (0.60) CCR1KCNH2ADRB1CYP3A4
SCHEMBL1671005 0.86 CCR1 (0.68) CCR1KCNH2ADRB1CYP3A4
SCHEMBL28797733 0.85 CCR1 (0.59) CCR1KCNH2ADRB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2491028-A1 INDAZOLE AND PYRAZOLOPYRIDINE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-08-29 EP disclosed
WO-2011049917-A1 INDAZOLE AND PYRAZOLOPYRIDINE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-04-28 WO disclosed