SCHEMBL1670957

SCHEMBL1670957

CCc1onc(C)c1-n1c(C(N)=NO)ccc1-c1ccc(O)cc1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.33
PIM1 P11309 5/20 0.33
CHEK1 O14757 3/20 0.32
CDK2 P24941 3/20 0.32
CSNK2A1 P68400 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670956 1.00 NTRK1 (0.33) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1672939 0.74 BRD4 (0.35)
SCHEMBL1672940 0.74 BRD4 (0.35)
SCHEMBL1670665 0.70 BRD4 (0.32) NTRK1PIM1
SCHEMBL1670663 0.70 BRD4 (0.32) NTRK1PIM1
SCHEMBL1670273 0.69 BRD4 (0.33) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1670272 0.69 BRD4 (0.33) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL1671278 0.65 BRD4 (0.33)
SCHEMBL1671281 0.65 BRD4 (0.33)
SCHEMBL1077888 0.63 ESR1 (0.36) NTRK1PIM1CHEK1CDK2CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed