SCHEMBL1671060

SCHEMBL1671060

O=C(O[C@@H]1CC[C@@H](c2cccc(F)c2F)C(O)c2cccnc21)N1CCC(n2c(=O)[nH]c3ncccc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 1.00
ADRB2 P07550 1/20 0.85
CYP3A4 P08684 1/20 0.85
RAMP1 O60894 1/20 0.53
CALCA P06881 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516458 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
SCHEMBL1670790 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
SCHEMBL30231460 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
SCHEMBL1670772 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
SCHEMBL30231391 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
SCHEMBL1670773 1.00 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
Rimegepant SCHEMBL24131009 0.92 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
Rimegepant SCHEMBL29374210 0.92 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
Rimegepant SCHEMBL2523699 0.92 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA
Rimegepant SCHEMBL29592766 0.92 CALCRL (1.00) CALCRLADRB2CYP3A4RAMP1CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488512-A1 CGRP RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2012-08-22 EP disclosed
WO-2011046997-A1 CGRP RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-04-21 WO disclosed