SCHEMBL16716631

SCHEMBL16716631

CCOC(=O)c1cn2ncnc(C)c2c1C

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 3/20 0.56
KDR P35968 9/20 0.53
MAPK14 Q16539 2/20 0.52
EGFR P00533 5/20 0.50
ERBB2 P04626 5/20 0.50
NR1H2 P55055 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1227597 0.87 MAP2K1 (0.55) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL1227820 0.86 KDR (0.60) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL1226304 0.86 MAP2K1 (0.54) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL32664156 0.76 MAP2K1 (0.50) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL4046095 0.76 EGFR (0.60) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL4044082 0.76 KDR (0.52) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL1730410 0.75 NR1H2 (0.73) MAP2K1KDRMAPK14NR1H2
SCHEMBL4102366 0.75 MAP2K1 (0.49) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL6112565 0.75 MAP2K1 (0.59) MAP2K1KDRMAPK14EGFRERBB2
SCHEMBL4101070 0.75 MAP2K1 (0.44) MAP2K1KDRMAPK14EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1497019-B1 PYRROLO-TRIAZINE ANILINE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2015-05-20 EP disclosed