SCHEMBL1672795

SCHEMBL1672795

CC(C)[Si](OC1CCC(c2cccc(F)c2F)C(O)c2cccnc21)(C(C)C)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 9/20 0.49
ADRB2 P07550 1/20 0.39
CYP3A4 P08684 1/20 0.39
HTR1A P08908 4/20 0.36
SLC6A2 P23975 4/20 0.36
SLC6A4 P31645 4/20 0.36
P2RX7 Q99572 6/20 0.35
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670184 1.00 CALCRL (0.49) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL16615981 1.00 CALCRL (0.49) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL830000 1.00 CALCRL (0.49) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL829734 1.00 CALCRL (0.49) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL16624591 0.88 CALCRL (0.38) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL16616000 0.88 CALCRL (0.38) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL16615999 0.88 CALCRL (0.38) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL15674334 0.87 CALCRL (0.48) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL1670444 0.87 CALCRL (0.38) CALCRLADRB2CYP3A4HTR1ASLC6A2
SCHEMBL15674335 0.87 CALCRL (0.48) CALCRLADRB2CYP3A4HTR1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488512-A1 CGRP RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2012-08-22 EP disclosed
WO-2011046997-A1 CGRP RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-04-21 WO disclosed