SCHEMBL16740698

SCHEMBL16740698

NC(=O)c1ccc(F)c(C(=O)c2c[nH]c3nccc(-c4ccc(Cl)cc4)c23)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.47
CYP3A4 P08684 9/20 0.47
KDR P35968 3/20 0.46
MAP2K2 P36507 3/20 0.46
MAP2K1 Q02750 3/20 0.46
MAP3K20 Q9NYL2 3/20 0.46
MAP4K5 Q9Y4K4 3/20 0.46
PLK4 O00444 2/20 0.46
MAP4K4 O95819 2/20 0.46
ABL1 P00519 2/20 0.46
FRK P42685 2/20 0.46
CDK8 P49336 2/20 0.46
CLK2 P49760 2/20 0.46
CSNK1G2 P78368 2/20 0.46
MINK1 Q8N4C8 2/20 0.46
HIPK4 Q8NE63 2/20 0.46
AURKB Q96GD4 2/20 0.46
SLK Q9H2G2 2/20 0.46
HIPK2 Q9H2X6 2/20 0.46
CDC7 O00311 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2888458 0.86 CYP3A4 (0.60) LRRK2CYP3A4KDRMAP2K2MAP2K1
SCHEMBL12520259 0.81 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19
SCHEMBL857622 0.81 MAP4K4 (0.63) LRRK2KDRMAP2K2MAP2K1MAP3K20
SCHEMBL4021568 0.80 LRRK2 (0.47) LRRK2CYP3A4KDRMAP2K2MAP2K1
SCHEMBL12521698 0.80 CYP3A4 (0.44) CYP3A4CYP2C9BRAFCYP2C19
SCHEMBL2888193 0.80 CYP3A4 (0.61) LRRK2CYP3A4CYP2C9BRAFCYP2C19
SCHEMBL857223 0.80 LRRK2 (0.52) LRRK2CYP3A4KDRMAP2K2MAP2K1
SCHEMBL3705714 0.79 CYP3A4 (0.51) CYP3A4CYP2C9BRAFCYP2C19
SCHEMBL2888690 0.79 CYP3A4 (0.61) CYP3A4CDK2CDK9CDK5CYP2C9
SCHEMBL857464 0.79 LRRK2 (0.48) LRRK2CYP3A4KDRMAP2K2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015075749-A1 NOVEL PROCESSES FOR THE PREPARATION OF VEMURAFENIB LAURUS LABS PRIVATE LIMITED (IN) 2015-05-28 WO disclosed