SCHEMBL16748610

SCHEMBL16748610

Cc1nc2ccc(F)cc2n1-c1nc(N)nc(Nc2ccc(OC(F)(F)F)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BMI1 P35226 5/20 0.49
CHRNA7 P36544 4/20 0.48
DHFR P00374 2/20 0.46
IDH1 O75874 6/20 0.43
GALR2 O43603 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
KCNH2 Q12809 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16748614 0.91 BMI1 (0.51) BMI1CHRNA7DHFRIDH1GALR2
SCHEMBL16748450 0.89 BMI1 (0.52) BMI1CHRNA7DHFRGALR2
SCHEMBL16748533 0.87 BMI1 (0.64) BMI1DHFRCTSSCTSK
SCHEMBL16748475 0.87 CHRNA7 (0.51) BMI1CHRNA7DHFRIDH1
SCHEMBL16748445 0.87 BMI1 (0.50) BMI1DHFR
SCHEMBL16748528 0.86 BMI1 (0.66) BMI1DHFRGALR2
SCHEMBL15747454 0.85 BMI1 (0.47) BMI1CHRNA7DHFRIDH1KCNH2
SCHEMBL16748613 0.85 BMI1 (0.48) BMI1DHFR
SCHEMBL16748437 0.85 BMI1 (0.48) BMI1DHFR
SCHEMBL16748587 0.83 BMI1 (0.47) BMI1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975878-B2 Substituted triazine BMI-1 inhibitors PTC THERAPEUTICS, INC. (US) 2018-05-22 US claimed
US-20160297798-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS PTC THERAPEUTICS, INC. 2016-10-13 US claimed
US-9975878-B2 Substituted triazine BMI-1 inhibitors PTC THERAPEUTICS, INC. (US) 2018-05-22 US disclosed
US-9975878-B2 Substituted triazine BMI-1 inhibitors PTC THERAPEUTICS, INC. (US) 2018-05-22 US disclosed
US-9975878-B2 Substituted triazine BMI-1 inhibitors PTC THERAPEUTICS, INC. (US) 2018-05-22 US disclosed
US-20160297798-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS PTC THERAPEUTICS, INC. 2016-10-13 US disclosed
US-20160297798-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS PTC THERAPEUTICS, INC. 2016-10-13 US disclosed
US-20160297798-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS PTC THERAPEUTICS, INC. 2016-10-13 US disclosed
WO-2015076801-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS PTC THERAPEUTICS, INC. (US) 2015-05-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160297798-A1 SUBSTITUTED TRIAZINE BMI-1 INHIBITORS BMI1, BAZ2A, BAZ2B BMI1 1/4885CHRNA7 4795/4885DHFR 4017/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.