SCHEMBL1675205

SCHEMBL1675205

c1nc(NCCc2c[nH]cn2)c2cc(-c3ccc4c(c3)OCO4)ccc2n1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 18/20 0.68
CLK1 P49759 12/20 0.68
DYRK1A Q13627 11/20 0.68
CLK2 P49760 10/20 0.68
DYRK1B Q9Y463 10/20 0.68
CLK3 P49761 7/20 0.66
CYP2D6 P10635 7/20 0.63
CYP2C19 P33261 7/20 0.63
CYP1A2 P05177 6/20 0.63
CYP3A4 P08684 6/20 0.63
ALDH1A1 P00352 4/20 0.63
HSD17B10 Q99714 4/20 0.63
KDM4E B2RXH2 2/20 0.63
MAPT P10636 2/20 0.63
HPGD P15428 2/20 0.63
MAPK1 P28482 4/20 0.60
LMNA P02545 3/20 0.60
CYP2C9 P11712 3/20 0.60
USP2 O75604 3/20 0.60
MEN1 O00255 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1675194 0.82 CLK1 (0.68) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675157 0.82 CLK4 (0.62) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675243 0.81 CLK1 (1.00) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675391 0.80 CLK4 (0.82) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675327 0.80 CLK4 (1.00) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675261 0.79 CLK4 (0.81) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675360 0.79 CLK4 (0.57) CLK4CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL1675305 0.78 CLK4 (0.62) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675362 0.78 CLK1 (0.82) CLK4CLK1DYRK1ACLK2DYRK1B
SCHEMBL1675044 0.77 CLK4 (0.51) CLK4DYRK1ACYP2D6CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO claimed
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO disclosed