SCHEMBL1675231

SCHEMBL1675231

Cn1cc2ccc(-c3ccc4ncnc(NCc5cccs5)c4c3)cc2n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 19/20 0.70
DYRK1A Q13627 9/20 0.67
CYP2D6 P10635 9/20 0.63
CYP2C19 P33261 9/20 0.63
LMNA P02545 8/20 0.63
CYP1A2 P05177 8/20 0.63
CYP3A4 P08684 8/20 0.63
ALDH1A1 P00352 7/20 0.63
HSD17B10 Q99714 5/20 0.63
HIF1A Q16665 5/20 0.63
USP2 O75604 5/20 0.63
CLK1 P49759 2/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
TSHR P16473 5/20 0.62
CYP2C9 P11712 5/20 0.62
MAPK1 P28482 5/20 0.62
KDM4E B2RXH2 2/20 0.62
MAPT P10636 2/20 0.62
HPGD P15428 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1675126 0.79 CLK4 (1.00) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675331 0.78 CLK4 (1.00) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675155 0.77 CLK4 (0.86) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL29594697 0.76 CLK4 (1.00) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675086 0.76 CLK4 (1.00) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675326 0.75 CLK4 (0.66) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675066 0.75 CLK4 (0.73) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675050 0.73 CLK4 (1.00) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL18895220 0.72 NPC1 (0.70) CLK4DYRK1ACYP2D6CYP2C19LMNA
SCHEMBL1675091 0.71 CLK4 (0.72) CLK4DYRK1ACYP2D6CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO claimed
WO-2011041655-A1 QUINAZOLIN-4-AMINE DERIVATIVES; AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-04-07 WO disclosed