Lysine

Lysine

SCHEMBL1675387

NCC(=O)O.NCCCC[C@H](N)C(=O)O.NCCCC[C@H](N)C(=O)O.O=C(O)[C@@H]1CCCN1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARDPTGS1PTGS2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Lysine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.53
DPP7 Q9UHL4 6/20 0.39
DPP4 P27487 4/20 0.39
DPP8 Q6V1X1 3/20 0.39
DPP9 Q86TI2 2/20 0.39
FAP Q12884 1/20 0.37
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
ARG1 P05089 3/20 0.36
ARG2 P78540 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lysine SCHEMBL21796038 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL3094553 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL22157986 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL3100126 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL6276264 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL1675447 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL16038745 1.00 GSR (0.53) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL23834597 0.96 GSR (0.57) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL11660661 0.96 GSR (0.57) GSRDPP7DPP4DPP8DPP9
Lysine SCHEMBL1696608 0.96 GSR (0.57) GSRDPP7DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9458197-B2 Elastin digest compositions and methods utilizing same HUMAN MATRIX SCIENCES, LLC (US) 2016-10-04 US disclosed
US-20150004184-A1 ELASTIN DIGEST COMPOSITIONS AND METHODS UTILIZING SAME NULASTIN, INC. 2015-01-01 US disclosed
US-8871707-B2 Elastin producing fibroblast formulations and methods of using the same HUMAN MATRIX SCIENCES, LLC (US) 2014-10-28 US disclosed
US-8828927-B2 Elastin digest compositions and methods utilizing same HUMAN MATRIX SCIENCES, LLC (US) 2014-09-09 US disclosed
US-20130295122-A1 ELASTIN DIGEST COMPOSITIONS AND METHODS UTILIZING SAME NULASTIN, INC. 2013-11-07 US disclosed
US-8461113-B2 Elastin digest compositions and methods utilizing same HUMAN MATRIX SCIENCES, LLC (US) 2013-06-11 US disclosed
US-20110081322-A1 ELASTIN PRODUCING FIBROBLAST FORMULATIONS AND METHODS OF USING THE SAME NULASTIN, INC. 2011-04-07 US disclosed
US-20090281044-A1 ELASTIN DIGEST COMPOSITIONS AND METHODS UTILIZING SAME NULASTIN, INC. 2009-11-12 US disclosed