SCHEMBL16762467

SCHEMBL16762467

CCCn1ccc(N)cc1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 2/20 0.41
ALOX15 P16050 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
PDE5A O76074 1/20 0.40
ACACB O00763 1/20 0.39
BRPF1 P55201 1/20 0.37
GRM2 Q14416 4/20 0.37
TYR P14679 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
GFER P55789 1/20 0.36
EGFR P00533 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PI4KA P42356 1/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20417808 0.89 ACACB (0.41) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL7764049 0.87 TLR8 (0.45) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL20417807 0.84 PIK3CD (0.47) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL3377603 0.81 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL15653625 0.80 ACACB (0.42) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL7954619 0.79 SMN1; SMN2 (0.39) SMN1; SMN2ALDH1A1ALOX15HTTATM
SCHEMBL17563249 0.78 TYR (0.41) ALDH1A1PDE5AACACBGRM2TYR
SCHEMBL2688931 0.78 ACACB (0.40) ALDH1A1HTTPDE5AACACBGRM2
SCHEMBL18186968 0.77 ACACB (0.39) PDE5AACACBGRM2TYRGAA
SCHEMBL256009 0.77 MAP2K2 (0.41) PDE5AACACBGRM2TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2507243-B1 SPIROINDOLINONE PYRROLIDINES HOFFMANN LA ROCHE (CH) 2015-06-10 EP claimed
WO-2018136634-A1 FUSED HETEROCYCLIC COMPOUNDS AS SELECTIVE BMP INHIBITORS VANDERBILT UNIVERSITY (US) 2018-07-26 WO disclosed
EP-2507243-B1 SPIROINDOLINONE PYRROLIDINES HOFFMANN LA ROCHE (CH) 2015-06-10 EP disclosed