SCHEMBL16768686

SCHEMBL16768686

C=C(NCCc1nccn1Cc1ccc(Cl)cc1)C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.47
HSP90B1 P14625 6/20 0.47
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KCNH2 Q12809 2/20 0.41
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
HSP90AB1 P08238 1/20 0.39
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16768667 0.91 HSP90AA1 (0.47) HSP90AA1HSP90B1LMNASMN1; SMN2
SCHEMBL16768665 0.89 HSP90AA1 (0.51) HSP90AA1HSP90B1SMN1; SMN2ADRB1HSP90AB1
SCHEMBL16768651 0.88 HSP90AA1 (0.46) HSP90AA1HSP90B1HSP90AB1BRD4
SCHEMBL16768673 0.87 HSP90B1 (0.51) HSP90AA1HSP90B1LMNAHSP90AB1
SCHEMBL16133646 0.86 HSP90B1 (0.53) HSP90AA1HSP90B1LMNASMN1; SMN2HSP90AB1
SCHEMBL16064999 0.84 HSP90AA1 (0.48) HSP90AA1HSP90B1LMNASMN1; SMN2KCNH2
SCHEMBL16768685 0.83 HSP90AA1 (0.50) HSP90AA1HSP90B1SMN1; SMN2HSP90AB1BRD4
SCHEMBL16136332 0.81 HSP90B1 (0.55) HSP90AA1HSP90B1LMNASMN1; SMN2HSP90AB1
SCHEMBL16133645 0.76 HSP90B1 (0.52) HSP90AA1HSP90B1LMNASMN1; SMN2
SCHEMBL16133633 0.76 HSP90B1 (0.49) HSP90AA1HSP90B1LMNASMN1; SMN2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9776996-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2017-10-03 US disclosed
US-9045477-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2015-06-02 US disclosed