SCHEMBL1679138

SCHEMBL1679138

C=CCC(C(=O)O)c1ccc(-c2ccc(O)cc2Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.52
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
ESR1 P03372 8/20 0.42
ESR2 Q92731 3/20 0.42
HCAR2 Q8TDS4 1/20 0.40
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
APP P05067 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
HSD17B10 Q99714 1/20 0.37
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
SRD5A2 P31213 1/20 0.35
FFAR2 O15552 1/20 0.35
DGAT1 O75907 1/20 0.35
SOAT1 P35610 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11077670 0.80 CYP2C19 (0.73) CYP2C19ESR1ESR2CYP3A4CYP2C9
SCHEMBL1679513 0.80 CYP2C19 (0.49) CYP2C19HSD17B1ESR1ESR2HCAR2
SCHEMBL1679476 0.80 CYP2C19 (0.59) CYP2C19AKR1C3AKR1C2APPCYP3A4
SCHEMBL1679465 0.76 CYP2C19 (0.44) CYP2C19HSD17B1ESR1ESR2AKR1C3
SCHEMBL21561158 0.76 CYP2C19 (0.71) CYP2C19CYP3A4CYP2C9HSD17B10FFAR2
SCHEMBL19803299 0.76 CYP2C19 (0.71) CYP2C19CYP3A4CYP2C9HSD17B10FFAR2
SCHEMBL4029220 0.76 CYP2C19 (0.71) CYP2C19CYP3A4CYP2C9HSD17B10FFAR2
SCHEMBL5879216 0.75 CYP2C19 (0.60) CYP2C19AKR1C3AKR1C2FFAR2
SCHEMBL624052 0.75 CYP2C19 (0.60) CYP2C19AKR1C3AKR1C2FFAR2
SCHEMBL5879212 0.75 CYP2C19 (0.60) CYP2C19AKR1C3AKR1C2FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7923573-B2 Benzene compound having 2 or more substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-04-12 US disclosed