SCHEMBL16800396

SCHEMBL16800396

Cc1cc(-n2cncn2)cnc1CC(=O)N1CCN(CCc2ccc3c(c2)COC3=O)CC1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 18/20 0.61
KCNJ1 P48048 17/20 0.61
SLC6A4 P31645 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4549776 0.89 KCNH2 (0.78) KCNH2KCNJ1SLC6A4
SCHEMBL15196864 0.87 KCNH2 (0.79) KCNH2KCNJ1SLC6A4
SCHEMBL15196879 0.85 KCNH2 (0.80) KCNH2KCNJ1
SCHEMBL15196818 0.85 KCNH2 (0.63) KCNH2KCNJ1SLC6A4
SCHEMBL15196936 0.83 KCNH2 (0.72) KCNH2KCNJ1SLC6A4
SCHEMBL15196846 0.83 KCNJ1 (0.78) KCNH2KCNJ1SLC6A4
SCHEMBL15196881 0.81 KCNH2 (0.65) KCNH2KCNJ1SLC6A4
SCHEMBL15196883 0.81 KCNJ1 (0.65) KCNH2KCNJ1SLC6A4
SCHEMBL15196958 0.81 KCNH2 (0.62) KCNH2KCNJ1SLC6A4
SCHEMBL15196820 0.79 KCNJ1 (0.64) KCNH2KCNJ1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9056859-B2 Inhibitors of the renal outer medullary potassium channel MERCK SHARP & DOHME CORP. (US) 2015-06-16 US disclosed