SCHEMBL16804244

SCHEMBL16804244

CCN1CCC(c2ccnc3c2ccn3Cc2ccc(C(N)=O)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
GAA P10253 1/20 0.40
CCNT1 O60563 2/20 0.38
CDK9 P50750 2/20 0.38
KLKB1 P03952 1/20 0.37
CNR1 P21554 1/20 0.36
FGFR1 P11362 1/20 0.36
FGFR4 P22455 1/20 0.36
NAMPT P43490 1/20 0.36
SCN9A Q15858 4/20 0.36
KCNH2 Q12809 2/20 0.36
SCN5A Q14524 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
DRD2 P14416 1/20 0.35
HTR6 P50406 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18108939 0.79 HDAC6 (0.57) KCNH2HDAC4HDAC1HDAC6
SCHEMBL18108920 0.79 HDAC6 (0.45) KCNH2HDAC4HDAC1HDAC6
SCHEMBL16804420 0.79 KDM4E (0.43) CNR1SCN9AKCNH2SCN5AOPRD1
SCHEMBL16804352 0.79 KDM4E (0.41) KCNH2OPRD1OPRK1
SCHEMBL16804034 0.79 KDM4E (0.46) OPRM1HDAC1
SCHEMBL18108847 0.79 CHKA (0.51) GAACNR1SCN9AKCNH2SCN5A
SCHEMBL18852715 0.78 CHKA (0.43) CCNT1CDK9FGFR1FGFR4OPRD1
SCHEMBL16804049 0.78 HDAC6 (0.46) KCNH2HDAC4HDAC1HDAC6
SCHEMBL18125622 0.78 HDAC6 (0.55) SCN9AKCNH2SCN5AHDAC4HDAC1
SCHEMBL16804320 0.78 KDM4E (0.41) FGFR1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015087151-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2015-06-18 WO disclosed