SCHEMBL16857656

SCHEMBL16857656

COc1cnc(OC(=O)Nc2ccc(F)c([C@]3(C)CO[C@@](C)(C(F)(F)F)C(N)=N3)c2)c(Cl)c1

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.73
BACE2 Q9Y5Z0 16/20 0.70
APP P05067 12/20 0.70
CYP2D6 P10635 6/20 0.70
CYP3A4 P08684 5/20 0.66
CYP2C9 P11712 2/20 0.66
CTSD P07339 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16857633 1.00 BACE1 (0.73) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857615 0.95 BACE1 (0.65) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857655 0.95 BACE1 (0.65) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857666 0.92 BACE1 (0.79) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857607 0.92 BACE1 (0.79) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857594 0.90 BACE1 (0.65) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857611 0.90 BACE1 (0.65) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857593 0.89 BACE1 (0.72) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857647 0.89 BACE1 (0.64) BACE1BACE2APPCYP2D6CYP3A4
SCHEMBL16857648 0.89 BACE1 (0.64) BACE1BACE2APPCYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2663559-B1 OXAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS NOVARTIS AG (CH) 2015-07-01 EP claimed