SCHEMBL16880980

SCHEMBL16880980

O=C(O)c1cncc(Cc2ccc(CO)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.49
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
DDO Q99489 1/20 0.44
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
HTT P42858 1/20 0.40
GFER P55789 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
SRD5A2 P31213 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318665 0.86 MEN1 (0.52) HCAR2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL7817677 0.86 HCAR2 (0.59) HCAR2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL30777432 0.86 HCAR2 (0.59) HCAR2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL7937454 0.80 SAE1 (0.47) CYP11B1CYP11B2ALDH1A1KDM4EMEN1
SCHEMBL3317267 0.80 MKNK1 (0.64) HCAR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL16881310 0.79 KMT2A (0.60) HCAR2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL16880864 0.79 CYP2C9 (0.56) ALDH1A1POLBCYP2C9CYP2C19HTT
SCHEMBL16881474 0.79 RECQL (0.49) CYP11B1CYP11B2ALDH1A1KDM4EMEN1
SCHEMBL16880732 0.78 CYP17A1 (0.40) CYP11B1CYP11B2POLBCYP2C9CYP2C19
SCHEMBL16891355 0.78 HSD17B3 (0.42) CYP11B1CYP11B2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3089746-A1 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2016-11-09 EP disclosed
WO-2015103317-A1 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2015-07-09 WO disclosed