SCHEMBL1689169

SCHEMBL1689169

CN(C)C(=O)C(C(=O)Nc1ccccc1)c1ccc(C(=O)Nc2cc(-c3ccccc3)ccc2N)cc1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.64
HDAC2 Q92769 9/20 0.61
HDAC3 O15379 3/20 0.61
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2108411 0.91 HDAC1 (0.74) HDAC1HDAC2HDAC3
SCHEMBL1689203 0.91 HDAC1 (0.60) HDAC1HDAC2HDAC3
SCHEMBL1689174 0.89 HDAC1 (0.67) HDAC1HDAC2HDAC3
SCHEMBL1689363 0.87 HDAC1 (0.82) HDAC1HDAC2HDAC3
SCHEMBL2107623 0.84 HDAC1 (0.68) HDAC1HDAC2HDAC3
SCHEMBL1689223 0.83 HDAC1 (0.71) HDAC1HDAC2HDAC3
SCHEMBL2108793 0.82 HDAC2 (0.65) HDAC1HDAC2HDAC3
SCHEMBL1689215 0.81 HDAC2 (0.75) HDAC1HDAC2HDAC3
SCHEMBL1689148 0.80 HDAC1 (0.59) HDAC1HDAC2HDAC3KCNH2
SCHEMBL18653509 0.79 HDAC2 (0.75) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-B1 MODIFIED MALONATE DERIVATIVES MERCK SHARP & DOHME (US) 2015-07-15 EP claimed
US-8158825-B2 Modified malonate derivatives MERCK SHARP & DOHME CORP. (US) 2012-04-17 US claimed
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP claimed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO claimed
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed