SCHEMBL16893085

SCHEMBL16893085

Cc1cnc(Nc2cccc(OCc3ccccc3)c2)nc1-c1c[nH]c(OC(=O)NC(CO)c2ccccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AURKA O14965 18/20 0.62
CDK2 P24941 16/20 0.62
MAPK1 P28482 9/20 0.62
MAP3K7 O43318 1/20 0.48
FLT3 P36888 1/20 0.48
GSK3A P49840 1/20 0.48
MAPK10 P53779 1/20 0.48
ROCK1 Q13464 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16892996 0.93 AURKA (0.64) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16892999 0.92 AURKA (0.64) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893070 0.90 AURKA (0.66) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893089 0.90 AURKA (0.75) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893123 0.88 AURKA (0.65) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893053 0.87 AURKA (0.66) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893003 0.87 AURKA (0.64) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16892980 0.86 AURKA (0.65) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893115 0.86 AURKA (0.67) AURKACDK2MAPK1MAP3K7FLT3
SCHEMBL16893049 0.86 AURKA (0.63) AURKACDK2MAPK1MAP3K7FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363906-B1 HETEROCYCLIC INHIBITORS OF ERK2 AND USES THEREOF VERTEX PHARMA (US) 2015-07-15 EP claimed