SCHEMBL16893108

SCHEMBL16893108

Nc1ncc(-c2cc(F)cc(C(F)(F)F)c2)c(-c2c[nH]c(OC(=O)NC(CO)c3ccccc3)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 10/20 0.42
ADORA1 P30542 2/20 0.42
ADORA2A P29274 1/20 0.42
AURKA O14965 7/20 0.40
CDK2 P24941 6/20 0.40
CDK5 Q00535 2/20 0.38
CDK5R1 Q15078 2/20 0.38
PDE2A O00408 1/20 0.36
CLK1 P49759 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16893090 0.85 AURKA (0.45) MAPK1ADORA1ADORA2AAURKACDK2
SCHEMBL16893098 0.80 AURKA (0.56) MAPK1AURKACDK2
SCHEMBL16893135 0.78 MAPK1 (0.43) MAPK1AURKACDK2
SCHEMBL5401943 0.75 ADORA1 (0.47) ADORA1ADORA2ACDK5CDK5R1CLK1
SCHEMBL16893029 0.74 AURKA (0.48) MAPK1AURKACDK2
SCHEMBL16892979 0.73 MAPK1 (0.58) MAPK1AURKACDK2
SCHEMBL16893049 0.72 AURKA (0.63) MAPK1AURKACDK2
SCHEMBL16893148 0.72 MAPK1 (0.78) MAPK1AURKACDK2
SCHEMBL16893137 0.72 MAPK1 (0.46) MAPK1AURKACDK2
SCHEMBL16893021 0.71 MAPK1 (0.57) MAPK1AURKACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363906-B1 HETEROCYCLIC INHIBITORS OF ERK2 AND USES THEREOF VERTEX PHARMA (US) 2015-07-15 EP claimed