SCHEMBL16900331

SCHEMBL16900331

CCc1ccc(N)cc1[C@@]1(C)N=C(N)COCC1(F)F

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.47
BACE2 Q9Y5Z0 9/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2593133 0.84 BACE1 (0.63) BACE1BACE2
SCHEMBL2592658 0.84 BACE1 (0.63) BACE1BACE2
SCHEMBL16900330 0.82 BACE1 (0.48) BACE1BACE2
Formic Acid SCHEMBL14759734 0.80 BACE1 (0.57) BACE1BACE2
SCHEMBL2589234 0.73 BACE1 (0.57) BACE1BACE2
SCHEMBL2589230 0.73 BACE1 (0.57) BACE1BACE2
SCHEMBL12478872 0.73 BACE1 (0.56) BACE1BACE2
SCHEMBL12478871 0.73 BACE1 (0.56) BACE1BACE2
SCHEMBL2593010 0.72 BACE1 (0.64) BACE1BACE2
SCHEMBL2592791 0.72 BACE1 (0.64) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9079919-B2 Spiro-[1,3]-oxazines and spiro-[1,4]-oxazepines as BACE1 and/or BACE2 inhibitors HOFFMANN-LA ROCHE INC. (US) 2015-07-14 US disclosed