SCHEMBL16938043

SCHEMBL16938043

Cc1ccc(-c2nc(-c3cc(N)ncn3)sc2-c2ncc[nH]2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.43
CCNE1 P24864 3/20 0.43
CDK2 P24941 3/20 0.43
DBF4 Q9UBU7 3/20 0.43
ROCK1 Q13464 1/20 0.36
KMO O15229 1/20 0.35
CCNT1 O60563 2/20 0.34
CSNK2A2 P19784 2/20 0.34
CSNK1A1 P48729 2/20 0.34
CSNK1D P48730 2/20 0.34
CDK9 P50750 2/20 0.34
CSNK2B P67870 2/20 0.34
CSNK2A1 P68400 2/20 0.34
NISCH Q9Y2I1 1/20 0.33
PIK3R2 O00459 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
JAK2 O60674 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6842885 0.91 CDC7 (0.42) CDC7CCNE1CDK2DBF4ROCK1
SCHEMBL16938035 0.85 CDC7 (0.42) CDC7CCNE1CDK2DBF4ROCK1
SCHEMBL16938037 0.82 CDC7 (0.41) CDC7CCNE1CDK2DBF4CCNT1
SCHEMBL16938045 0.78 ROCK1 (0.44) CDC7CCNE1CDK2DBF4ROCK1
SCHEMBL6842852 0.76 CDC7 (0.43) CDC7CCNE1CDK2DBF4ROCK1
SCHEMBL6842851 0.75 CDC7 (0.40) CDC7CCNE1CDK2DBF4CCNT1
SCHEMBL16938044 0.74 CDC7 (0.38) CDC7CCNE1CDK2DBF4ROCK1
SCHEMBL17089258 0.72 CDC7 (0.33) CDC7CCNE1CDK2DBF4NISCH
SCHEMBL16938046 0.72 CDC7 (0.36) CDC7CCNE1CDK2DBF4PIK3CD
SCHEMBL17089259 0.71 JAK2 (0.36) ROCK1CSNK1A1CDK9NISCHJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9090601-B2 Thiazole derivatives MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-07-28 US disclosed