SCHEMBL16972727

SCHEMBL16972727

CCc1c(-c2ccc(-c3cn[nH]c3)cc2)[nH]c(=O)c2c(=O)[nH]sc12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.51
ACVR1 Q04771 1/20 0.35
PDE10A Q9Y233 1/20 0.34
AKT2 P31751 2/20 0.34
AKT1 P31749 1/20 0.34
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
XDH P47989 1/20 0.33
ROCK2 O75116 7/20 0.33
PDE7A Q13946 1/20 0.33
PRKCQ Q04759 1/20 0.33
TNIK Q9UKE5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972674 0.80 KCNH2 (0.47) KCNH2ACVR1ROCK2PRKCQ
SCHEMBL16984188 0.76 KCNH2 (0.52) KCNH2
SCHEMBL16984186 0.71 KCNH2 (0.50) KCNH2
SCHEMBL16972695 0.68 KCNH2 (0.61) KCNH2
SCHEMBL16984192 0.67 KCNH2 (0.40) KCNH2
SCHEMBL16984191 0.67 KCNH2 (0.72) KCNH2
SCHEMBL16972673 0.66 KCNH2 (0.66) KCNH2
SCHEMBL7895370 0.64 AKT2 (0.59) AKT2AKT1ROCK2
SCHEMBL16432987 0.63 AKT2 (0.76) ACVR1AKT2AKT1ROCK2PRKCQ
SCHEMBL15689115 0.63 AKT2 (0.76) ACVR1AKT2AKT1ROCK2PRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed