SCHEMBL16972737

SCHEMBL16972737

CCOC(=O)c1c(O)c(CC)c(-c2ccc(N3CCC(N(C)C)C3)cc2)[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.59
MCHR1 Q99705 8/20 0.41
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
CLK2 P49760 1/20 0.39
MAP4K2 Q12851 1/20 0.39
CAMK2D Q13557 1/20 0.39
DYRK1A Q13627 1/20 0.39
PIM3 Q86V86 1/20 0.39
AURKB Q96GD4 1/20 0.39
PRKD2 Q9BZL6 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
STK17A Q9UEE5 1/20 0.39
MAP4K5 Q9Y4K4 1/20 0.39
TLR9 Q9NR96 3/20 0.39
TLR7 Q9NYK1 3/20 0.39
TLR8 Q9NR97 2/20 0.39
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14758924 0.89 KCNH2 (0.62) KCNH2MCHR1TLR9TLR7TLR8
Hydrochloric Acid SCHEMBL14745204 0.88 KCNH2 (0.61) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL14741162 0.77 KCNH2 (0.48) KCNH2MCHR1
SCHEMBL14741145 0.76 KCNH2 (0.46) KCNH2MCHR1PRKD3MAP4K4PIM1
SCHEMBL14741188 0.76 KCNH2 (0.46) KCNH2
SCHEMBL16577241 0.76 KCNH2 (0.46) KCNH2
SCHEMBL14745170 0.76 KCNH2 (0.46) KCNH2
SCHEMBL14745169 0.76 KCNH2 (0.47) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL16568257 0.75 TP53 (0.55) CYP1A2CYP2C19LMNA
SCHEMBL14741044 0.75 KCNH2 (0.46) KCNH2MCHR1PRKD3MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed