SCHEMBL16986792

SCHEMBL16986792

COc1ccc(-c2nn3c(-c4cnc(N5CCN(OC(=O)OC(C)(C)C)CC5)nc4)cnc3s2)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.54
FYN P06241 5/20 0.42
KDM4E B2RXH2 3/20 0.41
MAPK1 P28482 3/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 2/20 0.41
LMNA P02545 2/20 0.41
USP2 O75604 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
DCTPP1 Q9H773 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CFTR P13569 1/20 0.40
HPGD P15428 2/20 0.39
HIF1A Q16665 1/20 0.39
SMPD3 Q9NY59 1/20 0.39
SIRT1 Q96EB6 1/20 0.38
KDM4C Q9H3R0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532196 0.88 PIK3CA (0.55) PIK3CAFYNKDM4EMAPK1ALDH1A1
SCHEMBL533182 0.83 PIK3CA (0.71) PIK3CAFYNKDM4EMAPK1ALDH1A1
SCHEMBL16986790 0.83 PIK3CA (0.68) PIK3CAFYNKDM4EALDH1A1CFTR
SCHEMBL532217 0.80 PIK3CA (0.64) PIK3CAFYNKDM4EMAPK1ALDH1A1
SCHEMBL532633 0.75 PIK3CA (0.74) PIK3CAFYNKDM4EMAPK1ALDH1A1
SCHEMBL2121133 0.75 PIK3CA (0.77) PIK3CAFYNCFTRSMPD3
SCHEMBL15975820 0.73 PIK3CA (0.59) PIK3CAFYNCFTRSMPD3
SCHEMBL532197 0.73 SMPD3 (0.49) PIK3CAKDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL533110 0.73 PIK3CA (0.70) PIK3CAFYNCFTRSMPD3
SCHEMBL532289 0.72 PIK3CA (0.67) PIK3CAFYNKDM4EMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414369-B1 IMIDAZO[2,1-B][1,3,4]THIADIAZOLE DERIVATIVES FUNDACIÓN CT NAC DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (ES) 2015-08-12 EP claimed