SCHEMBL17004692

SCHEMBL17004692

CCCCc1cc2ncc(C#Cc3ccc(C)cc3)cn2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KIT P10721 4/20 0.38
DDR1 Q08345 3/20 0.38
GRM5 P41594 1/20 0.37
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
KCNH2 Q12809 2/20 0.32
MAPT P10636 2/20 0.31
NOS2 P35228 1/20 0.31
DDR2 Q16832 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1992121 0.79 NPC1 (0.61) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1991109 0.77 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL9903131 0.69 KIT (0.56) KITDDR1GRM5DDR2
SCHEMBL1990467 0.69 NPC1 (0.48) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1993210 0.69 NPC1 (0.63) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1992598 0.68 NPC1 (0.50) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1996110 0.67 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1990294 0.67 EGLN1 (0.39) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1991532 0.67 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNAKDM4E
SCHEMBL1995378 0.67 APP (0.38) NPC1RAB9ASMN1; SMN2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513102-B1 ETHYNYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2015-08-19 EP disclosed