SCHEMBL17019555

SCHEMBL17019555

CCc1c(N)ncnc1N1CCC(c2nc(-c3ccc(F)c(C)c3)cn2CCN)CC1

nearest known ligand 0.85

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 20/20 0.85
AKT1 P31749 20/20 0.85
AKT2 P31751 2/20 0.69
KCNH2 Q12809 2/20 0.69
AKT3 Q9Y243 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16247301 0.92 RPS6KB1 (1.00) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL16987133 0.92 RPS6KB1 (0.97) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL14792364 0.92 RPS6KB1 (1.00) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL14791635 0.92 RPS6KB1 (0.87) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL16247302 0.91 RPS6KB1 (1.00) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL14792365 0.91 RPS6KB1 (0.79) RPS6KB1AKT1
SCHEMBL16247265 0.91 RPS6KB1 (0.86) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL16247266 0.91 RPS6KB1 (0.88) RPS6KB1AKT1
SCHEMBL16247267 0.90 RPS6KB1 (0.84) RPS6KB1AKT1AKT2KCNH2AKT3
SCHEMBL14792251 0.90 RPS6KB1 (1.00) RPS6KB1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015123174-A1 PYRIMIDINE IMIDAZOLE AMINES AS MODULATORS OF KINASE ACTIVITY MERCK PATENT GMBH (DE) 2015-08-20 WO disclosed