SCHEMBL17022907

SCHEMBL17022907

CCc1nnc2c(C(F)(F)F)c(CN[C@H]3CC[C@@H](c4ccccc4)CC3)ccn12

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.63
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SLC6A3 Q01959 1/20 0.50
SIGMAR1 Q99720 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4561619 1.00 GRM2 (0.63) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4561618 1.00 GRM2 (0.63) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL5019350 0.90 GRM2 (0.58) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4560523 0.90 GRM2 (0.54) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4561583 0.90 GRM2 (0.54) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4560522 0.90 GRM2 (0.54) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4561653 0.89 GRM2 (0.73) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4562065 0.89 GRM2 (0.73) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL4561654 0.89 GRM2 (0.73) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1
SCHEMBL10322385 0.84 GRM2 (0.80) GRM2CYP2C9CYP2C19SLC6A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649069-B1 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS JANSSEN PHARMACEUTICALS INC (US) 2015-08-26 EP claimed