SCHEMBL17028064

SCHEMBL17028064

Cc1cc(C(F)(F)F)cnc1N[C@H]1CCCC1NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.58
HDAC4 P56524 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HCRTR2 O43614 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17007122 1.00 HCRTR1 (0.58) HCRTR1HDAC4HDAC6HCRTR2
SCHEMBL22131260 0.90 HCRTR1 (0.57) HCRTR1HDAC4HDAC6HCRTR2
SCHEMBL17007392 0.90 HCRTR1 (0.57) HCRTR1HDAC4HDAC6HCRTR2
SCHEMBL17007268 0.89 HCRTR1 (0.58) HCRTR1
SCHEMBL22131257 0.89 HCRTR1 (0.58) HCRTR1
SCHEMBL17007180 0.89 HCRTR1 (0.56) HCRTR1HDAC4HDAC6HCRTR2
SCHEMBL17017351 0.87 HCRTR1 (0.44) HCRTR1HDAC4HDAC6
SCHEMBL17007191 0.86 HCRTR1 (0.64) HCRTR1
SCHEMBL17007313 0.81 HCRTR1 (0.59) HCRTR1HDAC4HDAC6HCRTR2
SCHEMBL17017349 0.81 HCRTR1 (0.43) HCRTR1HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107898-A1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS Takeda Pharmaceutical Company Limited (JP) 2016-12-28 EP disclosed
WO-2015124932-A1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA CAMBRIDGE LIMITED (GB) 2015-08-27 WO disclosed